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Istradefylline forty mg/day greater peak ranges and AUC of CYP3A4 substrates in scientific trials. This effect was not observed with istradefylline 20 mg/working day. Take into account dose reduction of sensitive CYP3A4 substrates.fluconazole will enhance the stage or impact of diazepam by affecting hepatic/intestinal enzyme CYP3A4 metabolism. Use